3
Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T16670 | PS210 | PDK | |
PS210 is a potent and selective activator of PDK1 (Kd: 3 μM), specifically targeting the PIF-binding pocket of PDK1, without acting against other protein kinases such as S6K, PKB/Akt, or GSK3. Its prodrug, PS423, serves ... | |||
T12639 | (R)-PS210 | Others | |
(R)-PS210, the R enantiomer of PS210 is a substrate-selective allosteric PDK1 activator with an (AC50 of 1.8 μM). | |||
T24676 | PS423 | PS210AM,PS 210 AM,PS 423,PS210-AM,PS-423 | |
PS423 is a substrate-selective protein kinase PDK1 inhibitor that acts by binding to the PIF-pocket allosteric docking site. |